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Publication : Developing EZH2-Targeted Therapy for Lung Cancer.

First Author  Frankel AE Year  2016
Journal  Cancer Discov Volume  6
Issue  9 Pages  949-52
PubMed ID  27587466 Mgi Jnum  J:236869
Mgi Id  MGI:5810025 Doi  10.1158/2159-8290.CD-16-0800
Citation  Frankel AE, et al. (2016) Developing EZH2-Targeted Therapy for Lung Cancer. Cancer Discov 6(9):949-52
abstractText  Epigenetic targets are exciting new avenues for cancer drug discovery. Zhang and colleagues have designed the open-source EZH2 inhibitor JQEZ5 and shown antitumor efficacy in vitro and in vivo in preclinical studies in murine and human lung adenocarcinoma models expressing high levels of EZH2. Cancer Discov; 6(9); 949-52. (c)2016 AACRSee related article by Zhang and colleagues, p. 1006.
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